X-ray structure of 1-deoxy-D-xylulose 5-phosphate reductoisomerase, DXR, Rv2870c, from Mycobacterium tuberculosis, in complex with manganese.
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X-ray structure of 1-deoxy-D-xylulose 5-phosphate reductoisomerase, DXR, Rv2870c, from Mycobacterium tuberculosis, in complex with manganese. Descriptor: 1-DEOXY-D-XYLULOSE 5-PHOSPHATE REDUCTOISOMERASE, MANGANESE (II) ION Authors: Henriksson, L.M, Larsson, A.M.S, Bergfors, T, Bjorkelid, C, Unge, T, Mowbray, S.L, Jones, T.A. Deposit date: 2010-12-08 Release date: 2011-06-29 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Design, Synthesis and X-Ray Crystallographic Studies of Alpha-Aryl Substituted Fosmidomycin Analogues as Inhibitors of Mycobacterium Tuberculosis 1-Deoxy-D-Xylulose-5-Phosphate Reductoisomerase J.Med.Chem, 54, 2011
结核分枝杆菌(Mycobacterium tuberculosis)来源的1-脱氧-D-木酮糖5-磷酸还原异构酶(1-deoxy-D-xylulose 5-phosphate reductoisomerase,简称DXR,基因标识Rv2870c)与锰离子形成复合物的X射线晶体结构。结构描述符:1-脱氧-D-木酮糖5-磷酸还原异构酶、锰(II)离子。作者:Henriksson, L.M.、Larsson, A.M.S.、Bergfors, T.、Björkelid, C.、Unge, T.、Mowbray, S.L.、Jones, T.A.。提交日期:2010年12月8日;发布日期:2011年6月29日;最后修改日期:2023年12月20日。实验方法:X射线衍射(分辨率1.9埃)。引用文献:《α-芳基取代膦霉素类似物的设计、合成及X射线晶体学研究——作为结核分枝杆菌1-脱氧-D-木酮糖5-磷酸还原异构酶抑制剂》,《药物化学杂志》(J.Med.Chem),2011年,第54卷。
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2010-12-08



