five

DHNA complex with 2-Amino-5-bromo-3-hydroxy-6-phenylpyrimidine

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Protein Data Bank Japan2024-02-14 更新2026-03-21 收录
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DHNA complex with 2-Amino-5-bromo-3-hydroxy-6-phenylpyrimidine Descriptor: 2-AMINO-5-BROMO-6-PHENYLPYRIMIDIN-4-OL, Dihydroneopterin aldolase Authors: Sanders, W.J, Nienaber, V.L, Lerner, C.G, McCall, J.O, Merrick, S.M, Swanson, S.J, Harlan, J.E, Stoll, V.S, Stamper, G.F, Betz, S.F, Condroski, K.R, Meadows, R.P, Severin, J.M, Walter, K.A, Magdalinos, P, Jakob, C.G, Wagner, R, Beutel, B.A. Deposit date: 2003-12-09 Release date: 2004-03-30 Last modified: 2024-02-14 Method: X-RAY DIFFRACTION (2.2 Å) Cite: Discovery of Potent Inhibitors of Dihydroneopterin Aldolase Using CrystaLEAD High-Throughput X-ray Crystallographic Screening and Structure-Directed Lead Optimization. J.Med.Chem., 47, 2004
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2003-12-09
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