five

Structure of Aurora A mutant bound to Biogenidec cpd 15

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Protein Data Bank Japan2024-02-28 更新2026-03-21 收录
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Structure of Aurora A mutant bound to Biogenidec cpd 15 Descriptor: 7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1H-pyrrol-3-yl}amino)-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamide, Aurora kinase A, MAGNESIUM ION, ... Authors: Silvian, L, Marcotte, D.J. Deposit date: 2012-01-27 Release date: 2012-07-18 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (2.8 Å) Cite: Structure-based design of 2,6,7-trisubstituted-7H-pyrrolo[2,3-d]pyrimidines as Aurora kinases inhibitors. Bioorg.Med.Chem.Lett., 22, 2012
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2012-01-27
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