rat LDHA in complex with 2-((3,4-dimethoxyphenyl)methyl))propanedioic acid
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rat LDHA in complex with 2-((3,4-dimethoxyphenyl)methyl))propanedioic acid Descriptor: 2-((3,4-DIMETHOXYPHENYL)METHYL))PROPANEDIOIC ACID, L-LACTATE DEHYDROGENASE A CHAIN Authors: Tucker, J.A, Brassington, C, Hassall, G, Vogtherr, M, Ward, R, Tart, J, Davies, G, Debreczeni, J. Deposit date: 2012-02-16 Release date: 2012-03-21 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (1.93 Å) Cite: The Design and Synthesis of Novel Lactate Dehydrogenase a Inhibitors by Fragment-Based Lead Generation J.Med.Chem., 55, 2012
大鼠乳酸脱氢酶A(LDHA)与2-((3,4-二甲氧基苯基)甲基)丙二酸的复合物
配体描述:2-((3,4-二甲氧基苯基)甲基)丙二酸、L-乳酸脱氢酶A亚基
作者:Tucker, J.A、Brassington, C、Hassall, G、Vogtherr, M、Ward, R、Tart, J、Davies, G、Debreczeni, J.
提交日期:2012-02-16
发布日期:2012-03-21
末次修改日期:2024-05-01
实验方法:X射线衍射(分辨率1.93埃)
引用文献:《基于片段导向先导化合物发现的新型乳酸脱氢酶A抑制剂的设计与合成》,《药物化学杂志》(J.Med.Chem.),第55卷,2012年
创建时间:
2012-02-16



