five

17beta-HSD5 in complex with 3,6-dihydropyridin-1(2H)-yl(5-methyl-1H-indol-2-yl)methanone

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Protein Data Bank Japan2024-05-29 更新2026-03-21 收录
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17beta-HSD5 in complex with 3,6-dihydropyridin-1(2H)-yl(5-methyl-1H-indol-2-yl)methanone Descriptor: 3,6-dihydropyridin-1(2H)-yl(5-methyl-1H-indol-2-yl)methanone, Aldo-keto reductase family 1 member C3, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE Authors: Amano, Y, Yamaguchi, T. Deposit date: 2014-09-09 Release date: 2015-04-15 Last modified: 2024-05-29 Method: X-RAY DIFFRACTION (1.94 Å) Cite: Structures of complexes of type 5 17 beta-hydroxysteroid dehydrogenase with structurally diverse inhibitors: insights into the conformational changes upon inhibitor binding. Acta Crystallogr.,Sect.D, 71, 2015

17β-羟基类固醇脱氢酶5型(17beta-HSD5)与3,6-二氢吡啶-1(2H)-基(5-甲基-1H-吲哚-2-基)甲酮的复合物 描述项:3,6-二氢吡啶-1(2H)-基(5-甲基-1H-吲哚-2-基)甲酮、醛酮还原酶家族1成员C3(Aldo-keto reductase family 1 member C3)、烟酰胺腺嘌呤二核苷酸磷酸(NADP, NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE) 作者:Amano Y、Yamaguchi T 存档日期:2014-09-09 发布日期:2015-04-15 最后修改日期:2024-05-29 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率1.94埃(Å) 引用文献:5型17β-羟基类固醇脱氢酶与结构多样抑制剂的复合物结构:抑制剂结合后的构象变化洞察. Acta Crystallogr.,Sect.D, 71, 2015
创建时间:
2014-09-09
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