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N-terminal expression tag remainder of human Carbonic Anhydrase II covalently modified by fragment

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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N-terminal expression tag remainder of human Carbonic Anhydrase II covalently modified by fragment Descriptor: (4-CARBOXYPHENYL)(CHLORO)MERCURY, 1-(1,3-dimethyl-1H-pyrazol-5-yl)methanamine, Carbonic anhydrase 2, ... Authors: Gloeckner, S, Heine, A, Klebe, G. Deposit date: 2019-07-16 Release date: 2020-04-15 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (1.02 Å) Cite: A Proof-of-Concept Fragment Screening of a Hit-Validated 96-Compounds Library against Human Carbonic Anhydrase II. Biomolecules, 10, 2020

经片段描述符共价修饰的人碳酸酐酶II(Carbonic Anhydrase II)的N端表达标签残留片段,涉及的片段描述符包括:(4-羧基苯基)(氯)汞、1-(1,3-二甲基-1H-吡唑-5-基)甲胺、碳酸酐酶2等。作者:Gloeckner S、Heine A、Klebe G。沉积日期:2019-07-16;发布日期:2020-04-15;最后修改日期:2024-11-06。实验方法:X射线衍射(X-RAY DIFFRACTION,分辨率1.02 Å)。引用文献:《针对人碳酸酐酶II的经命中验证的96种化合物库片段筛选概念验证研究》,刊载于《生物分子》(Biomolecules),2020年,第10卷。
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2019-07-16
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