ephB4 kinase domain inhibitor complex
收藏Protein Data Bank Japan2023-12-13 更新2026-03-21 收录
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https://pdbj.org/mine/summary/2vwx
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ephB4 kinase domain inhibitor complex Descriptor: 3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzenesulfonamide, EPHRIN TYPE-B RECEPTOR 4, MAGNESIUM ION Authors: Read, J, Brassington, C.A, Green, I, McCall, E.J, Valentine, A.L, Barratt, D, Leach, A.G, Kettle, J.G. Deposit date: 2008-06-27 Release date: 2008-10-28 Last modified: 2023-12-13 Method: X-RAY DIFFRACTION (1.65 Å) Cite: Inhibitors of the Tyrosine Kinase Ephb4. Part 2: Structure-Based Discovery and Optimisation of 3,5-Bis Substituted Anilinopyrimidines. Bioorg.Med.Chem.Lett., 18, 2008
创建时间:
2008-06-27



