Crystal structure of TRIM24 with 3,4-dimethoxy-N-(6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)benzenesulfonamide inhibitor
收藏Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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Crystal structure of TRIM24 with 3,4-dimethoxy-N-(6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)benzenesulfonamide inhibitor Descriptor: 3,4-dimethoxy-N-[6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl]benzenesulfonamide, DIMETHYL SULFOXIDE, PENTAETHYLENE GLYCOL, ... Authors: Tallant, C, Structural Genomics Consortium (SGC), Clark, P.G.K, Vieira, L.C.C, Krojer, T, Nunez-Alonso, G, Picaud, S, Fedorov, O, Dixon, D.J, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Brennan, P.E, Knapp, S. Deposit date: 2015-05-10 Release date: 2015-06-17 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (1.79 Å) Cite: Crystal structure of TRIM24 with 3,4-dimethoxy-N-(6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)benzenesulfonamide inhibitor To Be Published
结合3,4-二甲氧基-N-[6-(4-甲氧基苯氧基)-1,3-二甲基-2-氧代-2,3-二氢-1H-苯并[d]咪唑-5-基]苯磺酰胺抑制剂的TRIM24晶体结构
描述物:3,4-二甲氧基-N-[6-(4-甲氧基苯氧基)-1,3-二甲基-2-氧代-2,3-二氢-1H-苯并[d]咪唑-5-基]苯磺酰胺、二甲基亚砜(Dimethyl Sulfoxide)、五甘醇(Pentaethylene Glycol)等
作者:Tallant, C(结构基因组学联盟,SGC)、Clark, P.G.K、Vieira, L.C.C、Krojer, T、Nunez-Alonso, G、Picaud, S、Fedorov, O、Dixon, D.J、von Delft, F、Arrowsmith, C.H、Edwards, A.M、Bountra, C、Brennan, P.E、Knapp, S
提交日期:2015-05-10
发布日期:2015-06-17
最后修改日期:2024-01-10
实验方法:X射线衍射(1.79 Å)
引用说明:结合3,4-二甲氧基-N-(6-(4-甲氧基苯氧基)-1,3-二甲基-2-氧代-2,3-二氢-1H-苯并[d]咪唑-5-基)苯磺酰胺抑制剂的TRIM24晶体结构,待发表
创建时间:
2015-05-10



