Crystal structure of the inactive unphosphorylated IRAK4 kinase domain bound to AMP-PNP
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Crystal structure of the inactive unphosphorylated IRAK4 kinase domain bound to AMP-PNP Descriptor: Interleukin-1 receptor-associated kinase 4, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ... Authors: Ferrao, R, Wu, H. Deposit date: 2018-08-19 Release date: 2019-02-13 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.61 Å) Cite: Conformational flexibility and inhibitor binding to unphosphorylated interleukin-1 receptor-associated kinase 4 (IRAK4). J.Biol.Chem., 294, 2019
与AMP-PNP结合的非活化未磷酸化IRAK4激酶结构域的晶体结构
描述符:白介素1受体相关激酶4 (Interleukin-1 receptor-associated kinase 4, IRAK4)、镁离子(MAGNESIUM ION)、磷氨膦酸腺苷酯(PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER)……
作者:Ferrao R、Wu H
提交日期:2018-08-19
发布日期:2019-02-13
最后修改日期:2024-03-13
实验方法:X射线衍射(X-RAY DIFFRACTION,分辨率2.61埃)
引用文献:《未磷酸化白介素1受体相关激酶4(IRAK4)的构象灵活性与抑制剂结合》,发表于《生物化学杂志(Journal of Biological Chemistry)》,2019年,第294卷
创建时间:
2018-08-19



