CRYSTAL STRUCTURE OF PROTEIN TYROSINE PHOSPHATASE 1B COMPLEXED WITH 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID
收藏Protein Data Bank Japan2023-08-09 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/1c88
下载链接
链接失效反馈官方服务:
资源简介:
CRYSTAL STRUCTURE OF PROTEIN TYROSINE PHOSPHATASE 1B COMPLEXED WITH 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID Descriptor: 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID, PROTEIN (PROTEIN-TYROSINE PHOSPHATASE 1B) Authors: Iversen, L.F, Andersen, H.S, Mortensen, S.B, Moller, N.P. Deposit date: 2000-04-16 Release date: 2000-05-03 Last modified: 2023-08-09 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Structure-based design of a low molecular weight, nonphosphorus, nonpeptide, and highly selective inhibitor of protein-tyrosine phosphatase 1B. J.Biol.Chem., 275, 2000
与2-(草酰氨基)-4,5,6,7-四氢噻吩并[2,3-c]吡啶-3-羧酸结合的蛋白酪氨酸磷酸酶1B(Protein Tyrosine Phosphatase 1B)晶体结构
描述项:2-(草酰氨基)-4,5,6,7-四氢噻吩并[2,3-c]吡啶-3-羧酸、蛋白质(蛋白酪氨酸磷酸酶1B)
作者:Iversen L.F.、Andersen H.S.、Mortensen S.B.、Møller N.P.
提交日期:2000-04-16
发布日期:2000-05-03
最后修改日期:2023-08-09
实验方法:X射线衍射(分辨率1.8 Å)
引用文献:基于结构设计的蛋白酪氨酸磷酸酶1B低分子量、非磷、非肽类高选择性抑制剂。《生物化学杂志》,275卷,2000年
创建时间:
2000-04-16



