Selection of fragments for kinase inhibitor design: decoration is key
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Selection of fragments for kinase inhibitor design: decoration is key Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6H)-one, SULFATE ION, ... Authors: Czodrowski, P, Hoelzemann, G, Barnickel, G, Greiner, H, Musil, D. Deposit date: 2014-11-26 Release date: 2015-08-12 Last modified: 2026-03-04 Method: X-RAY DIFFRACTION (1.51 Å) Cite: Selection of fragments for kinase inhibitor design: decoration is key. J.Med.Chem., 58, 2015
激酶抑制剂设计的片段筛选:修饰是关键
描述符:2-氨基-2-羟甲基-1,3-丙二醇、4-[(4-氨基苯基)氨基]吡啶并[2,3-d]嘧啶-5(6H)-酮、硫酸根离子……
作者:Czodrowski P、Hoelzemann G、Barnickel G、Greiner H、Musil D
提交日期:2014-11-26
发布日期:2015-08-12
最后修改日期:2026-03-04
检测方法:X射线衍射(1.51 Å)
引用文献:《激酶抑制剂设计的片段筛选:修饰是关键》,J.Med.Chem.,第58卷,2015年
创建时间:
2014-11-26



