Wild Type HIV-1 Protease with Antiviral Drug Saquinavir
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Wild Type HIV-1 Protease with Antiviral Drug Saquinavir Descriptor: (2S)-N-[(2S,3R)-4-[(2S,3S,4aS,8aS)-3-(tert-butylcarbamoyl)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-hydroxy-1 -phenyl-butan-2-yl]-2-(quinolin-2-ylcarbonylamino)butanediamide, FORMIC ACID, Protease, ... Authors: Kovalevsky, A.Y, Wang, Y.-F, Tie, Y, Weber, I.T. Deposit date: 2010-09-21 Release date: 2010-11-10 Last modified: 2023-09-06 Method: X-RAY DIFFRACTION (1.16 Å) Cite: Atomic resolution crystal structures of HIV-1 protease and mutants V82A and I84V with saquinavir Proteins, 67, 2007
携带抗病毒药物沙奎那韦(Saquinavir)的野生型HIV-1蛋白酶。描述物:(2S)-N-[(2S,3R)-4-[(2S,3S,4aS,8aS)-3-(叔丁基甲酰氨基)-3,4,4a,5,6,7,8,8a-八氢-1H-异喹啉-2-基]-3-羟基-1-苯基丁-2-基]-2-(喹啉-2-基羰基氨基)丁二酰胺、甲酸(FORMIC ACID)、蛋白酶(Protease)等;作者:Kovalevsky, A.Y、Wang, Y.-F、Tie, Y、Weber, I.T.;存放日期:2010-09-21;发布日期:2010-11-10;最后修改日期:2023-09-06;实验方法:X射线衍射(X-RAY DIFFRACTION,分辨率1.16埃(Å));引用文献:《HIV-1蛋白酶及其突变体V82A与I84V结合沙奎那韦的原子分辨率晶体结构》,《Proteins》,第67卷,2007年
创建时间:
2010-09-21



