five

Modulation of MLL1 Methyltransferase Activity

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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Modulation of MLL1 Methyltransferase Activity Descriptor: (2~{S})-2-[[(2~{S})-2-[[(2~{S})-2-azanyl-3-oxidanyl-propanoyl]amino]propanoyl]amino]-5-carbamimidamido-~{N}-[(2~{S})-1-[[4-[(~{E})-[4-(hydroxymethyl)phenyl]diazenyl]phenyl]methylamino]-1-oxidanylidene-propan-2-yl]pentanamide, WD repeat-containing protein 5 Authors: Srinivasan, V. Deposit date: 2016-10-11 Release date: 2017-06-28 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (2.43 Å) Cite: Controlled inhibition of methyltransferases using photoswitchable peptidomimetics: towards an epigenetic regulation of leukemia. Chem Sci, 8, 2017
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2016-10-11
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