Crystal structure of SETDB1 Tudor domain with aryl triazole fragments
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Crystal structure of SETDB1 Tudor domain with aryl triazole fragments Descriptor: 1,2-ETHANEDIOL, Histone-lysine N-methyltransferase SETDB1, N-{[2-(3,5-dimethyl-4H-1,2,4-triazol-4-yl)phenyl]methyl}acetamide, ... Authors: MADER, P, Mendoza-Sanchez, R, IQBAL, A, DONG, A, DOBROVETSKY, E, CORLESS, V.B, LIEW, S.K, TEMPEL, W, SMIL, D, DELA SENA, C.C, KENNEDY, S, DIAZ, D, HOLOWNIA, A, VEDADI, M, BROWN, P.J, SANTHAKUMAR, V, Bountra, C, Edwards, A.M, YUDIN, A.K, Arrowsmith, C.H, Structural Genomics Consortium (SGC) Deposit date: 2017-08-30 Release date: 2017-09-27 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Crystal structure of SETDB1 Tudor domain with aryl triazole fragments to be published
结合芳基三唑片段的SETDB1 Tudor结构域晶体结构
描述符:1,2-乙二醇、组蛋白赖氨酸N-甲基转移酶SETDB1、N-{[2-(3,5-二甲基-4H-1,2,4-三唑-4-基)苯基]甲基}乙酰胺,……
作者:MADER, P、MENDOZA-SANCHEZ, R、IQBAL, A、DONG, A、DOBROVETSKY, E、CORLESS, V.B、LIEW, S.K、TEMPEL, W、SMIL, D、DE LA SENA, C.C、KENNEDY, S、DIAZ, D、HOLOWNIA, A、VEDADI, M、BROWN, P.J、SANTHAKUMAR, V、BOUNTRA, C、EDWARDS, A.M、YUDIN, A.K、ARROWSMITH, C.H、结构基因组学联合体(Structural Genomics Consortium, SGC)
提交日期:2017-08-30
发布日期:2017-09-27
最后修改日期:2024-03-13
实验方法:X射线衍射(分辨率1.8 Å)
引用说明:结合芳基三唑片段的SETDB1 Tudor结构域晶体结构(待发表)
创建时间:
2017-08-30



