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Crystal Structure of the Androgen Receptor Ligand Binding Domain with DHT and a peptide derived from its physiological coactivator GRIP1 NR box3

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Protein Data Bank Japan2024-02-14 更新2026-03-21 收录
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Crystal Structure of the Androgen Receptor Ligand Binding Domain with DHT and a peptide derived from its physiological coactivator GRIP1 NR box3 Descriptor: 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, Nuclear receptor coactivator 2 Authors: Estebanez-Perpina, E, Moore, J.M.R, Mar, E, Nguyen, P, Delgado-Rodrigues, E, Baxter, J.D, Webb, P, Fletterick, R.J, Guy, R.K. Deposit date: 2004-05-05 Release date: 2005-01-25 Last modified: 2024-02-14 Method: X-RAY DIFFRACTION (2.07 Å) Cite: The Molecular Mechanisms of Coactivator Utilization in Ligand-dependent Transactivation by the Androgen Receptor. J.Biol.Chem., 280, 2005

雄激素受体(Androgen Receptor)配体结合域结合5α-双氢睾酮(5-ALPHA-DIHYDROTESTOSTERONE,DHT)及源自其生理共激活因子GRIP1 NR box3的肽段的晶体结构 描述项:5α-双氢睾酮、雄激素受体、核受体共激活因子2(Nuclear receptor coactivator 2) 作者:Estebanez-Perpina, E、Moore, J.M.R、Mar, E、Nguyen, P、Delgado-Rodrigues, E、Baxter, J.D、Webb, P、Fletterick, R.J、Guy, R.K. 存放日期:2004-05-05 发布日期:2005-01-25 最后修改日期:2024-02-14 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率2.07埃(Å) 引用文献:《雄激素受体介导配体依赖性转录激活过程中共激活因子利用的分子机制》,《生物化学杂志》(J.Biol.Chem.),第280卷,2005年
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2004-05-05
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