COMPLEX OF THE CATALYTIC PORTION OF HUMAN HMG-COA REDUCTASE WITH CERIVASTATIN
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COMPLEX OF THE CATALYTIC PORTION OF HUMAN HMG-COA REDUCTASE WITH CERIVASTATIN Descriptor: 7-[4-(4-FLUORO-PHENYL)-5-HYDROXYMETHYL-2,6-DIISOPROPYL-PYRIDIN-3-YL]-3,5-DIHYDROXY-HEPTANOIC ACID, ADENOSINE-5'-DIPHOSPHATE, HMG-COA REDUCTASE Authors: Istvan, E.S, Deisenhofer, J. Deposit date: 2001-01-09 Release date: 2001-05-11 Last modified: 2023-08-09 Method: X-RAY DIFFRACTION (2.26 Å) Cite: Structural mechanism for statin inhibition of HMG-CoA reductase. Science, 292, 2001
人源羟甲基戊二酰辅酶A还原酶(HMG-CoA reductase催化域与西立伐他汀(cerivastatin)复合物
描述符:7-[4-(4-氟苯基)-5-羟甲基-2,6-二异丙基吡啶-3-基]-3,5-二羟基庚酸、腺苷-5'-二磷酸、羟甲基戊二酰辅酶A还原酶
作者:Istvan, E.S.、Deisenhofer, J.
存入日期:2001-01-09
发布日期:2001-05-11
最后修改日期:2023-08-09
实验方法:X射线衍射(2.26埃)
引用文献:他汀类药物抑制羟甲基戊二酰辅酶A还原酶的结构机制,《科学》,292卷,2001年。
创建时间:
2001-01-09



