CRYSTAL STRUCTURE OF HUMAN FKBP51 FK1 DOMAIN A19T MUTANT IN COMPLEX WITH NICOTINAMIDE
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CRYSTAL STRUCTURE OF HUMAN FKBP51 FK1 DOMAIN A19T MUTANT IN COMPLEX WITH NICOTINAMIDE Descriptor: CHLORIDE ION, NICOTINAMIDE, Peptidyl-prolyl cis-trans isomerase FKBP5, ... Authors: Fiegen, D, Draxler, S.W. Deposit date: 2020-01-13 Release date: 2020-05-27 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (0.98 Å) Cite: Hybrid Screening Approach for Very Small Fragments: X-ray and Computational Screening on FKBP51. J.Med.Chem., 63, 2020
人FKBP51 FK1结构域A19T突变体与烟酰胺复合物的晶体结构
描述项:氯离子、烟酰胺、肽基脯氨酰顺反异构酶FKBP5(Peptidyl-prolyl cis-trans isomerase FKBP5)等
作者:Fiegen, D.、Draxler, S.W.
存库日期:2020-01-13
发布日期:2020-05-27
最后更新日期:2024-01-24
实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率0.98 Å
引用:《针对超小片段的混合筛选策略:FKBP51的X射线与计算筛选》,《Journal of Medicinal Chemistry》(J.Med.Chem.),2020年,第63卷
创建时间:
2020-01-13



