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PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5010894431- (S,S) isomer

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Protein Data Bank Japan2023-09-20 更新2026-03-21 收录
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PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5010894431- (S,S) isomer Descriptor: (1S,2S)-1-[2-chloro-4-(cyclopropylcarbamamido)benzamido]-4-hydroxy-2,3-dihydro-1H-indene-2-carboxylic acid, Non-structural protein 3 Authors: Correy, G.J, Fraser, J.S. Deposit date: 2022-06-09 Release date: 2022-07-06 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (1.05 Å) Cite: Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023

PanDDA分析小组提交数据集——新型冠状病毒(SARS-CoV-2)NSP3宏结构域与Z5010894431-(S,S)异构体复合物的晶体结构。描述项:(1S,2S)-1-[2-氯-4-(环丙基甲酰氨基)苯甲酰氨基]-4-羟基-2,3-二氢-1H-茚-2-羧酸;靶蛋白:非结构蛋白3(Non-structural protein 3)。作者:Correy, G.J.、Fraser, J.S.。提交日期:2022-06-09,发布日期:2022-07-06,最后修改日期:2023-09-20。实验方法:X射线衍射(分辨率1.05 Å)。引用文献:《迭代计算设计与晶体筛选鉴定靶向新冠病毒Nsp3宏结构域的强效抑制剂》,《美国国家科学院院刊》,120卷,2023年
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2022-06-09
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