Crystal structure of the human CDK7 kinase domain in complex with LDC4297
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Crystal structure of the human CDK7 kinase domain in complex with LDC4297 Descriptor: 2-[(3R)-piperidin-3-yl]oxy-8-propan-2-yl-N-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amine, Cyclin-dependent kinase 7, GLYCEROL, ... Authors: Laursen, M, Caing-Carlsson, R, Houssari, R, Javadi, A, Kimbung, Y.R, Murina, V, Orozco-Rodriguez, J.M, Svensson, A, Welin, M, Logan, D, Svensson, B, Walse, B. Deposit date: 2023-05-23 Release date: 2023-06-14 Last modified: 2024-02-07 Method: X-RAY DIFFRACTION (2.75 Å) Cite: Crystal structure of the human CDK7 kinase domain in complex with LDC4297 To Be Published
人类CDK7激酶结构域与LDC4297复合物的晶体结构 描述:2-[(3R)-哌啶-3-基]氧基-8-异丙基-N-[(2-吡唑-1-基苯基)甲基]吡唑并[1,5-a][1,3,5]三嗪-4-胺、细胞周期蛋白依赖性激酶7(Cyclin-dependent kinase 7)、甘油(GLYCEROL)等 作者:Laursen M、Caing-Carlsson R、Houssari R、Javadi A、Kimbung Y.R、Murina V、Orozco-Rodriguez J.M、Svensson A、Welin M、Logan D、Svensson B、Walse B 沉积日期:2023-05-23 发布日期:2023-06-14 最后修改日期:2024-02-07 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率2.75 Å 引用信息:人类CDK7激酶结构域与LDC4297复合物的晶体结构 [待发表]



