PARP15 catalytic domain in complex with OUL220
收藏Protein Data Bank Japan2024-01-31 更新2026-03-28 收录
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https://pdbj.org/mine/summary/7ouw
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PARP15 catalytic domain in complex with OUL220 Descriptor: 8-methoxy-4~{H}-thieno[2,3-c]isoquinolin-5-one, DIMETHYL SULFOXIDE, Protein mono-ADP-ribosyltransferase PARP15 Authors: Maksimainen, M.M, Lehtio, L. Deposit date: 2021-06-14 Release date: 2021-12-08 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.6 Å) Cite: Analogs of TIQ-A as inhibitors of human mono-ADP-ribosylating PARPs. Bioorg.Med.Chem., 52, 2021
PARP15催化结构域与OUL220复合物 描述:8-甲氧基-4H-噻吩并[2,3-c]异喹啉-5-酮、二甲基亚砜、蛋白质单ADP核糖基转移酶PARP15
作者:Maksimainen, M.M.、Lehtio, L.
存储日期:2021-06-14
发布日期:2021-12-08
最后修改日期:2024-01-31
实验方法:X射线衍射(分辨率1.6 Å)
引用文献:《TIQ-A类似物作为人类单ADP核糖基化PARPs的抑制剂》,Bioorg.Med.Chem., 52, 2021
创建时间:
2021-06-14



