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LIGAND BINDING DOMAIN OF HUMAN PPAR-GAMMA IN COMPLEX WITH THE AGONIST PIOGLITAZONE

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Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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https://pdbj.org/mine/summary/2xkw
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LIGAND BINDING DOMAIN OF HUMAN PPAR-GAMMA IN COMPLEX WITH THE AGONIST PIOGLITAZONE Descriptor: (5R)-5-{4-[2-(5-ethylpyridin-2-yl)ethoxy]benzyl}-1,3-thiazolidine-2,4-dione, 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ... Authors: Mueller, J.J, Schupp, M, Unger, T, Kintscher, U, Heinemann, U. Deposit date: 2010-07-14 Release date: 2011-08-10 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (2.02 Å) Cite: Binding Diversity of Pioglitazone by Peroxisome Proliferator-Activated Receptor-Gamma To be Published

与人过氧化物酶体增殖物激活受体γ(Peroxisome Proliferator-Activated Receptor Gamma, PPAR-γ)配体结合域与激动剂吡格列酮(Pioglitazone)复合物 描述:(5R)-5-{4-[2-(5-乙基吡啶-2-基)乙氧基]苄基}-1,3-噻唑烷-2,4-二酮、2-{2-[2-(2-{2-[2-(2-乙氧基-乙氧基)-乙氧基]-乙氧基}-乙氧基)-乙氧基]-乙氧基}-乙醇、4-(2-羟乙基)-1-哌嗪乙磺酸等 作者:J.J. Mueller、M. Schupp、T. Unger、U. Kintscher、U. Heinemann 存入日期:2010-07-14 发布日期:2011-08-10 最后修改日期:2023-12-20 实验方法:X射线衍射(2.02 Å) 引用文献:《过氧化物酶体增殖物激活受体γ介导的吡格列酮结合多样性》(Binding Diversity of Pioglitazone by Peroxisome Proliferator-Activated Receptor-Gamma),待发表
创建时间:
2010-07-14
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