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Elaborate Manifold of Short Hydrogen Bond Arrays Mediating Binding of Active Site-Directed Serine Protease Inhibitors

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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Elaborate Manifold of Short Hydrogen Bond Arrays Mediating Binding of Active Site-Directed Serine Protease Inhibitors Descriptor: 3-{5-[AMINO(IMINIO)METHYL]-1H-INDOL-2-YL}-5-METHOXY-1,1'-BIPHENYL-2-OLATE, BETA-TRYPSIN, CALCIUM ION, ... Authors: Katz, B.A, Elrod, K, Verner, E, Mackman, R.L, Luong, C, Shrader, W.D, Sendzik, M, Spencer, J.R, Sprengeler, P.A, Kolesnikov, A, Tai, V.W, Hui, H.C, Breitenbucher, J.G, Allen, D, Janc, J.W. Deposit date: 2003-03-06 Release date: 2003-09-02 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.62 Å) Cite: Elaborate manifold of short hydrogen bond arrays mediating binding of active site-directed serine protease inhibitors. J.Mol.Biol., 329, 2003

介导活性位点靶向丝氨酸蛋白酶(serine protease)抑制剂结合的短氢键阵列(hydrogen bond array)精细调控网络 数据集描述符:3-{5-[氨基(亚胺鎓)甲基]-1H-吲哚-2-基}-5-甲氧基-1,1'-联苯-2-醇盐、β-胰蛋白酶(β-Trypsin)、钙离子(Calcium Ion)等 作者:Katz, B.A、Elrod, K、Verner, E、Mackman, R.L、Luong, C、Shrader, W.D、Sendzik, M、Spencer, J.R、Sprengeler, P.A、Kolesnikov, A、Tai, V.W、Hui, H.C、Breitenbucher, J.G、Allen, D、Janc, J.W 提交日期:2003-03-06 发布日期:2003-09-02 最后修改日期:2024-11-13 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率1.62埃(Å) 引用文献:介导活性位点靶向丝氨酸蛋白酶(serine protease)抑制剂结合的短氢键阵列(hydrogen bond array)精细调控网络. J.Mol.Biol., 329, 2003
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2003-03-06
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