THRb mutation with a novel agonist
收藏Protein Data Bank Japan2023-11-22 更新2026-03-21 收录
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THRb mutation with a novel agonist Descriptor: 2-[(1-methyl-4-oxidanyl-7-phenoxy-isoquinolin-3-yl)carbonylamino]ethanoic acid, Nuclear receptor coactivator 2, Thyroid hormone receptor beta Authors: Yao, B.Q, Li, Y. Deposit date: 2019-08-07 Release date: 2019-10-23 Last modified: 2023-11-22 Method: X-RAY DIFFRACTION (2.7 Å) Cite: Revealing a Mutant-Induced Receptor Allosteric Mechanism for the Thyroid Hormone Resistance. Iscience, 20, 2019
针对结合新型激动剂的甲状腺激素受体β(Thyroid hormone receptor beta,THRβ)突变体的数据集
描述符:2-[(1-甲基-4-羟基-7-苯氧基-异喹啉-3-基)羰基氨基]乙酸、核受体辅激活因子2(Nuclear receptor coactivator 2)、甲状腺激素受体β(Thyroid hormone receptor beta)
作者:Yao, B.Q、Li, Y.
提交日期:2019-08-07
发布日期:2019-10-23
最后修改日期:2023-11-22
研究方法:X射线衍射(X-RAY DIFFRACTION),分辨率2.7 Å
引用文献:《揭示甲状腺激素抵抗的突变诱导受体变构机制》,发表于《Iscience》第20卷,2019年
创建时间:
2019-08-07



