Crystal of Raucaffricine Glucosidase in complex with inhibitor

Crystal of Raucaffricine Glucosidase in complex with inhibitor Descriptor: (1R,2S,3S,4R,5R)-4-(cyclohexylmethylamino)-5-(hydroxymethyl)cyclopentane-1,2,3-triol, RAUCAFFRICINE-O-BETA-D-GLUCOSIDASE, SULFATE ION Authors: Xia, L, Lin, H, Panjikar, S, Ruppert, M, Castiglia, A, Rajendran, C, Wang, M, Schuebel, H, Warzecha, H, Jaeger, V, Stoeckigt, J. Deposit date: 2013-01-17 Release date: 2014-01-29 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Ligand Structures of Synthetic Deoxa-Pyranosylamines with Raucaffricine and Strictosidine Glucosidases Provide Structural Insights Into Their Binding and Inhibitory Behaviours. J.Enzyme.Inhib.Med.Chem., 30, 2015

劳卡弗辛葡糖苷酶（Raucaffricine Glucosidase）与抑制剂形成的复合物晶体
描述：(1R,2S,3S,4R,5R)-4-(环己基甲氨基)-5-(羟甲基)环戊烷-1,2,3-三醇、劳卡弗辛-O-β-D-葡糖苷酶、硫酸根离子
作者：Xia, L、Lin, H、Panjikar, S、Ruppert, M、Castiglia, A、Rajendran, C、Wang, M、Schuebel, H、Warzecha, H、Jaeger, V、Stoeckigt, J
入库日期：2013-01-17
发布日期：2014-01-29
最后更新日期：2023-12-20
实验方法：X射线衍射（X-RAY DIFFRACTION），分辨率2.4埃（Å）
引用文献：《合成脱氧吡喃胺类配体与劳卡弗辛葡糖苷酶和严格苷葡糖苷酶的结合结构及其结合与抑制行为的结构阐释》，刊载于《Journal of Enzyme Inhibition and Medicinal Chemistry》（缩写：J.Enzyme.Inhib.Med.Chem.），2015年，第30卷。