Overview of all used inhibitors.

NIAID Data Ecosystem2026-03-08 收录

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In general, we expect complete inhibition of the target at concentrations about 10 times above the IC50 value [38], [56].

创建时间：

2014-01-31

Crystal Structure of HSP90 with N-Aryl-benzimidazolone I

结构生物学

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Crystal Structure of HSP90 with N-Aryl-benzimidazolone I Descriptor: 1-(2,4-dihydroxyphenyl)-1,3-dihydro-2H-benzimidazol-2-one, Heat shock protein HSP 90-alpha Authors: Park, C.H. Deposit date: 2010-0

Protein Data Bank Japan2024-02-21 更新60

Mouse cGAS bound to the inhibitor RU365

药物靶点抑制

自身免疫疾病治疗

Mouse cGAS bound to the inhibitor RU365 Descriptor: (3R)-3-[1-(1H-benzimidazol-2-yl)-5-hydroxy-3-methyl-1H-pyrazol-4-yl]-2-benzofuran-1(3H)-one, Cyclic GMP-AMP synthase, DNA (5'-D(*AP*AP*AP*TP*TP*GP*C

Protein Data Bank Japan2024-05-22 更新40

Crystal structure of uPA in complex with upain-2-4-W3A

蛋白质晶体

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Crystal structure of uPA in complex with upain-2-4-W3A Descriptor: Urokinase-type plasminogen activator chain B, upain-2-4-W3A peptide Authors: Jiang, L, Huang, M. Deposit date: 2017-01-08 Release dat

Protein Data Bank Japan2024-10-16 更新40

Crystal structure of human Arginase-1 at pH 9.0 in complex with ABH

酶结构解析

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Crystal structure of human Arginase-1 at pH 9.0 in complex with ABH Descriptor: 2(S)-AMINO-6-BORONOHEXANOIC ACID, Arginase-1, MANGANESE (II) ION, ... Authors: Grobben, Y, Uitdehaag, J.C.M, Zaman, G.J.

Protein Data Bank Japan2024-01-24 更新50

Structure determination of a potent, selective antibody inhibitor of human MMP9 (apo MMP9)

蛋白质结构解析

药物靶点抑制

Structure determination of a potent, selective antibody inhibitor of human MMP9 (apo MMP9) Descriptor: CALCIUM ION, Matrix metalloproteinase-9,Matrix metalloproteinase-9, ZINC ION Authors: Appleby, T.

Protein Data Bank Japan2023-10-04 更新40

Overview of all used inhibitors.

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