Crystal Structure of BAZ2A bromodomain in complex with 1-methylpyridinone compound 5
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Crystal Structure of BAZ2A bromodomain in complex with 1-methylpyridinone compound 5 Descriptor: Bromodomain adjacent to zinc finger domain protein 2A, ~{N}-[3-[2-(dimethylamino)ethyl]-2-oxidanylidene-1,3-benzoxazol-5-yl]-1-methyl-6-oxidanylidene-pyridine-3-carboxamide Authors: Dalle Vedove, A, Spiliotopoulos, D, Lolli, G, Caflisch, A. Deposit date: 2018-01-10 Release date: 2018-05-30 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.1 Å) Cite: Structural Analysis of Small-Molecule Binding to the BAZ2A and BAZ2B Bromodomains. ChemMedChem, 13, 2018
BAZ2A溴结构域(bromodomain)与1-甲基吡啶酮化合物5复合物的晶体结构
描述:锌指结构域旁溴结构域蛋白2A(Bromodomain adjacent to zinc finger domain protein 2A, BAZ2A),N-[3-[2-(二甲基氨基)乙基]-2-氧代-1,3-苯并恶唑-5-基]-1-甲基-6-氧代吡啶-3-甲酰胺
作者:Dalle Vedove A、Spiliotopoulos D、Lolli G、Caflisch A
沉积日期:2018-01-10
发布日期:2018-05-30
最后修改日期:2024-01-17
实验方法:X射线衍射(1.1 Å)
引用:《小分子与BAZ2A及BAZ2B溴结构域结合的结构分析》,ChemMedChem,第13卷,2018年
创建时间:
2018-01-10



