Inhibition of cell-free MYC-MAX heterodimer formation and direct MYC binding*.

*Average IC50 values (μM) with standard deviation from the MYC-MAX ELISA and average KD values (μM) from the MYC SPR assay, as described in Experimental Procedures. IC50s and KDs of E, N, and C monomers alone are listed first, followed by IC50s and KDs from equimolar titrations of combinations of monomers. C11 and C12 are non-dimerizable control compounds corresponding to N11 and N12, respectively.Inhibition of cell-free MYC-MAX heterodimer formation and direct MYC binding*.