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The active form of a pentameric ion channel (sTeLIC) gated by alkaline pH - Co-crystallization with 4-bromo cinnamic acid

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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The active form of a pentameric ion channel (sTeLIC) gated by alkaline pH - Co-crystallization with 4-bromo cinnamic acid Descriptor: 3-(4-bromophenyl)propanoic acid, Cys-loop ligand-gated ion channel, nonyl beta-D-glucopyranoside Authors: Hu, H, Delarue, M. Deposit date: 2018-01-26 Release date: 2018-05-16 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (3 Å) Cite: Crystal structures of a pentameric ion channel gated by alkaline pH show a widely open pore and identify a cavity for modulation. Proc. Natl. Acad. Sci. U.S.A., 115, 2018

碱性pH门控的五聚体离子通道(sTeLIC)活性形式——与4-溴肉桂酸共结晶 描述项:3-(4-溴苯基)丙酸、半胱氨酸环配体门控离子通道(Cys-loop ligand-gated ion channel)、壬基β-D-吡喃葡萄糖苷(nonyl beta-D-glucopyranoside) 作者:Hu, H、Delarue, M 保藏日期:2018-01-26 发布日期:2018-05-16 最后更新:2024-05-08 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率3 Å 引用文献:碱性pH门控五聚体离子通道的晶体结构呈现广泛开放的孔道并鉴定出调控空腔,《美国国家科学院院刊》,2018年,第115卷
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2018-01-26
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