Crystal structure of ADAMTS5 with inhibitor bound
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Crystal structure of ADAMTS5 with inhibitor bound Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(N-HYDROXYAMINO)-2R-ISOBUTYL-2S-(2-THIENYLTHIOMETHYL)SUCCINYL-L-PHENYLALANINE-N-METHYLAMIDE, ADAMTS-5, ... Authors: Mosyak, L, Stahl, M, Somers, W. Deposit date: 2007-10-15 Release date: 2007-12-11 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Crystal structures of the two major aggrecan degrading enzymes, ADAMTS4 and ADAMTS5. Protein Sci., 17, 2008
结合抑制剂的ADAMTS5晶体结构
配体标识:2-乙酰氨基-2-脱氧-β-D-吡喃葡萄糖-(1→4)-2-乙酰氨基-2-脱氧-β-D-吡喃葡萄糖、4-(N-羟氨基)-2R-异丁基-2S-(2-噻吩硫甲基)琥珀酰-L-苯丙氨酸-N-甲基酰胺、ADAMTS-5……
作者:Mosyak, L、Stahl, M、Somers, W
沉积日期:2007-10-15
发布日期:2007-12-11
最后修改日期:2024-11-20
实验方法:X射线衍射(2.6 Å)
引用文献:《两种主要聚集蛋白聚糖降解酶ADAMTS4与ADAMTS5的晶体结构》,《Protein Science》,17卷,2008年
创建时间:
2007-10-15



