CYSTATHIONINE GAMMA-SYNTHASE IN COMPLEX WITH THE INHIBITOR APPA
收藏Protein Data Bank Japan2023-08-09 更新2026-03-21 收录
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CYSTATHIONINE GAMMA-SYNTHASE IN COMPLEX WITH THE INHIBITOR APPA Descriptor: 2-[(3-HYDROXY-2-METHYL-5-PHOSPHONOOXYMETHYL-PYRIDIN-4-YLMETHYL)-IMINO]-5-PHOSPHONO-PENT-3-ENOIC ACID, CYSTATHIONINE GAMMA-SYNTHASE Authors: Steegborn, C, Laber, B, Messerschmidt, A, Huber, R, Clausen, T. Deposit date: 2001-02-19 Release date: 2001-09-05 Last modified: 2023-08-09 Method: X-RAY DIFFRACTION (3.2 Å) Cite: Crystal structures of cystathionine gamma-synthase inhibitor complexes rationalize the increased affinity of a novel inhibitor. J.Mol.Biol., 311, 2001
胱硫醚γ合酶(cystathionine gamma-synthase)与抑制剂APPA的复合物
配体描述:2-[(3-羟基-2-甲基-5-膦酰氧基甲基-吡啶-4-基甲基)-亚氨基]-5-膦酰基-戊-3-烯酸(2-[(3-HYDROXY-2-METHYL-5-PHOSPHONOOXYMETHYL-PYRIDIN-4-YLMETHYL)-IMINO]-5-PHOSPHONO-PENT-3-ENOIC ACID)
作者:Steegborn, C、Laber, B、Messerschmidt, A、Huber, R、Clausen, T
提交日期:2001-02-19
发布日期:2001-09-05
最后修改日期:2023-08-09
实验方法:X射线衍射(X-RAY DIFFRACTION,3.2 Å)
引用文献:《胱硫醚γ合酶抑制剂复合物的晶体结构阐明了新型抑制剂的亲和力提升机制》,J.Mol.Biol., 311, 2001
创建时间:
2001-02-19



