Crystal Structure of HCK in complex with the fluorescent compound SKF86002
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Crystal Structure of HCK in complex with the fluorescent compound SKF86002 Descriptor: 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole, CALCIUM ION, CHLORIDE ION, ... Authors: Parker, L.J, Tanaka, A, Handa, N, Honda, K, Tomabechi, Y, Shirouzu, M, Yokoyama, S. Deposit date: 2013-07-25 Release date: 2014-02-12 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (2.85 Å) Cite: Kinase crystal identification and ATP-competitive inhibitor screening using the fluorescent ligand SKF86002. Acta Crystallogr.,Sect.D, 70, 2014
结合荧光化合物SKF86002的造血细胞激酶(HCK)晶体结构。描述符:6-(4-氟苯基)-5-(吡啶-4-基)-2,3-二氢咪唑并[2,1-b][1,3]噻唑、钙离子、氯离子…… 作者:Parker, L.J、Tanaka, A、Handa, N、Honda, K、Tomabechi, Y、Shirouzu, M、Yokoyama, S。提交日期:2013-07-25。发布日期:2014-02-12。最后修改日期:2024-10-30。实验方法:X射线衍射(2.85埃)。引用文献:使用荧光配体SKF86002进行激酶晶体鉴定与ATP竞争性抑制剂筛选。《Acta Crystallogr.,Sect.D》,70卷,2014年。
创建时间:
2013-07-25



