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The Catalytic Subunit of cAMP-dependent Protein Kinase (PKA) in Complex with Rho-kinase Inhibitor Y-27632

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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The Catalytic Subunit of cAMP-dependent Protein Kinase (PKA) in Complex with Rho-kinase Inhibitor Y-27632 Descriptor: (R)-TRANS-4-(1-AMINOETHYL)-N-(4-PYRIDYL) CYCLOHEXANECARBOXAMIDE, cAMP-dependent protein kinase inhibitor, alpha form, ... Authors: Breitenlechner, C, Gassel, M, Hidaka, H, Kinzel, V, Huber, R, Engh, R.A, Bossemeyer, D. Deposit date: 2003-08-22 Release date: 2003-12-16 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (2 Å) Cite: Protein kinase A in complex with Rho-kinase inhibitors Y-27632, Fasudil, and H-1152P: structural basis of selectivity. Structure, 11, 2003

与Rho激酶抑制剂Y-27632结合的cAMP依赖性蛋白激酶(cAMP-dependent Protein Kinase, PKA)催化亚基 数据集描述:(R)-反式-4-(1-氨乙基)-N-(4-吡啶基)环己烷甲酰胺,cAMP依赖性蛋白激酶抑制剂α型,…… 作者:Breitenlechner C、Gassel M、Hidaka H、Kinzel V、Huber R、Engh R.A、Bossemeyer D 保藏日期:2003-08-22 发布日期:2003-12-16 最后修订日期:2024-10-30 实验方法:X射线衍射(X-RAY DIFFRACTION,分辨率2 Å) 引用文献:结合Rho激酶抑制剂Y-27632、法舒地尔(Fasudil)与H-1152P的蛋白激酶A:选择性的结构基础。《Structure》,11卷,2003年
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2003-08-22
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