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XFEL crystal structure of human melatonin receptor MT1 in complex with 2-iodomelatonin

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Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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XFEL crystal structure of human melatonin receptor MT1 in complex with 2-iodomelatonin Descriptor: DI(HYDROXYETHYL)ETHER, GLYCEROL, N-[2-(2-iodo-5-methoxy-1H-indol-3-yl)ethyl]acetamide, ... Authors: Stauch, B, Johansson, L.C, McCorvy, J.D, Patel, N, Han, G.W, Gati, C, Batyuk, A, Ishchenko, A, Brehm, W, White, T.A, Michaelian, N, Madsen, C, Zhu, L, Grant, T.D, Grandner, J.M, Olsen, R.H.J, Tribo, A.R, Weierstall, U, Roth, B.L, Katritch, V, Liu, W, Cherezov, V. Deposit date: 2018-09-05 Release date: 2019-04-24 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (3.2 Å) Cite: Structural basis of ligand recognition at the human MT1melatonin receptor. Nature, 569, 2019

人类褪黑素受体MT1与2-碘褪黑素复合物的X射线自由电子激光(XFEL)晶体结构。 试剂清单:二(羟乙基)醚、甘油、N-[2-(2-碘-5-甲氧基-1H-吲哚-3-基)乙基]乙酰胺…… 作者:Stauch, B、Johansson, L.C、McCorvy, J.D、Patel, N、Han, G.W、Gati, C、Batyuk, A、Ishchenko, A、Brehm, W、White, T.A、Michaelian, N、Madsen, C、Zhu, L、Grant, T.D、Grandner, J.M、Olsen, R.H.J、Tribo, A.R、Weierstall, U、Roth, B.L、Katritch, V、Liu, W、Cherezov, V。 存档日期:2018-09-05;发布日期:2019-04-24;最后修改日期:2023-10-11。 实验方法:X射线衍射(分辨率3.2埃)。 引用文献:《人类MT1褪黑素受体配体识别的结构基础》,《自然》(*Nature*),第569卷,2019年
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2018-09-05
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