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PanDDA analysis group deposition -- Crystal Structure of Enterovirus D68 3C Protease in complex with Z57965168

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Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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https://pdbj.org/mine/summary/7gq8
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PanDDA analysis group deposition -- Crystal Structure of Enterovirus D68 3C Protease in complex with Z57965168 Descriptor: 4-[(difluoromethyl)sulfanyl]aniline, DIMETHYL SULFOXIDE, Protease 3C Authors: Lithgo, R.M, Fairhead, M, Koekemoer, L, Aschenbrenner, J.C, Balcomb, B.H, Godoy, A.S, Marples, P.G, Ni, X, Tomlinson, C.W.E, Thompson, W, Wild, C, Fearon, D, Walsh, M.A, von Delft, F. Deposit date: 2023-08-24 Release date: 2023-11-29 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (1.38 Å) Cite: Crystallographic Fragment Screen of Coxsackievirus A16 2A Protease identifies new opportunities for the development of broad-spectrum anti-enterovirals. Biorxiv, 2024

PanDDA分析团队提交的数据集——肠道病毒D68型3C蛋白酶与Z57965168复合物的晶体结构。描述组分:4-[(二氟甲基)硫基]苯胺、二甲基亚砜(DIMETHYL SULFOXIDE)、3C蛋白酶(Protease 3C)。作者:Lithgo, R.M、Fairhead, M、Koekemoer, L、Aschenbrenner, J.C、Balcomb, B.H、Godoy, A.S、Marples, P.G、Ni, X、Tomlinson, C.W.E、Thompson, W、Wild, C、Fearon, D、Walsh, M.A、von Delft, F。提交日期:2023-08-24;发布日期:2023-11-29;末次修改日期:2024-10-16。实验方法:X射线衍射(分辨率1.38埃)。引用文献:《柯萨奇病毒A16型2A蛋白酶晶体片段筛选发现广谱抗肠道病毒药物开发新方向》,BioRxiv,2024年
创建时间:
2023-08-24
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