Crystal structure of human MMP-7 in complex with inhibitor
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Crystal structure of human MMP-7 in complex with inhibitor Descriptor: CALCIUM ION, Matrilysin, Peptide Inhibitor, ... Authors: Kamitani, M, Oka, Y, Tabuse, H. Deposit date: 2022-02-15 Release date: 2022-10-05 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (1.5 Å) Cite: Discovery of Highly Potent and Selective Matrix Metalloproteinase-7 Inhibitors by Hybridizing the S1' Subsite Binder with Short Peptides. J.Med.Chem., 65, 2022
人基质金属蛋白酶-7(MMP-7)与抑制剂结合的晶体结构 描述项:钙离子(CALCIUM ION)、基质溶解素(Matrilysin)、肽类抑制剂(Peptide Inhibitor)等 作者:Kamitani, M、Oka, Y、Tabuse, H 沉积日期:2022-02-15 发布日期:2022-10-05 末次修改日期:2023-11-29 检测方法:X射线衍射(X-RAY DIFFRACTION),分辨率1.5埃(Å) 引用文献:《通过将S1'亚位点结合剂与短肽杂交发现高效且高选择性的基质金属蛋白酶-7抑制剂》,《药物化学杂志》(J.Med.Chem.),第65卷,2022年
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2022-02-15



