Mutant Imine Reductase IR007-143 from Amycolatopsis azurea, E120A, M197W, M206S, A213P, D238G, I240L
收藏Protein Data Bank Japan2026-03-04 更新2026-04-19 收录
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Mutant Imine Reductase IR007-143 from Amycolatopsis azurea, E120A, M197W, M206S, A213P, D238G, I240L Descriptor: Mutant Imine Reductase IR007-143 from Amycolatopsis azurea, E120A, M197W, ... Authors: Gilio, A.K, Grogan, G.J. Deposit date: 2022-11-08 Release date: 2023-09-20 Last modified: 2026-03-04 Method: X-RAY DIFFRACTION (2.7 Å) Cite: Engineering of a Reductive Aminase to Enable the Synthesis of a Key Intermediate to a CDK 2/4/6 Inhibitor Acs Catalysis, 13, 2023
本数据集的研究对象为源自天蓝马杜拉放线菌(Amycolatopsis azurea)的突变亚胺还原酶(Imine Reductase)IR007-143,其突变位点包括E120A、M197W、M206S、A213P、D238G、I240L。
描述:该突变亚胺还原酶IR007-143源自天蓝马杜拉放线菌(Amycolatopsis azurea),突变位点包括E120A、M197W……
作者:Gilio A.K.与Grogan G.J.
沉积日期:2022-11-08
发布日期:2023-09-20
最后修改日期:2026-03-04
实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率2.7埃
引用文献:《工程化还原胺化酶以合成CDK 2/4/6抑制剂(Cyclin-dependent kinase 2/4/6 inhibitor)关键中间体》,刊载于《ACS催化》,2023年,第13卷。
创建时间:
2022-11-08



