rat LDHA in complex with N-(2-(methylamino)-1,3-benzothiazol-6-yl) acetamide
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rat LDHA in complex with N-(2-(methylamino)-1,3-benzothiazol-6-yl) acetamide Descriptor: GLYCEROL, L-LACTATE DEHYDROGENASE A CHAIN, MALONATE ION, ... Authors: Tucker, J.A, Brassington, C, Hassall, G, Vogtherr, M, Ward, R, Tart, J, Davies, G, Greenwood, R. Deposit date: 2012-02-16 Release date: 2012-03-21 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (2.03 Å) Cite: The Design and Synthesis of Novel Lactate Dehydrogenase a Inhibitors by Fragment-Based Lead Generation J.Med.Chem., 55, 2012
大鼠LDHA与N-(2-(甲氨基)-1,3-苯并噻唑-6-基)乙酰胺的复合物
描述项:甘油、L-乳酸脱氢酶A链、丙二酸根离子……
作者:Tucker, J.A.、Brassington, C、Hassall, G、Vogtherr, M、Ward, R、Tart, J、Davies, G、Greenwood, R.
存档日期:2012-02-16
发布日期:2012-03-21
最后修改日期:2024-05-01
实验方法:X射线衍射(分辨率2.03埃)
引用文献:《基于片段先导物发现法设计并合成新型乳酸脱氢酶A抑制剂》,《药物化学杂志》(J.Med.Chem.),第55卷,2012年
创建时间:
2012-02-16



