Crystal Structure of MAPK7 (ERK5) with inhibitor
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Crystal Structure of MAPK7 (ERK5) with inhibitor Descriptor: 11-cyclopentyl-2-[[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl-phenyl]amino]-5-methyl-pyrimido[4,5-b][1,4]benzodiazepin-6-one, MITOGEN-ACTIVATED PROTEIN KINASE 7 Authors: Elkins, J.M, Wang, J, Vollmar, M, Mahajan, P, Savitsky, P, Deng, X, Gray, N.S, Pike, A.C.W, von Delft, F, Bountra, C, Arrowsmith, C, Edwards, A, Knapp, S. Deposit date: 2012-09-03 Release date: 2012-09-19 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (2.8 Å) Cite: X-Ray Crystal Structure of Erk5 (Mapk7) in Complex with a Specific Inhibitor. J.Med.Chem., 56, 2013
丝裂原活化蛋白激酶7(MAPK7,又称ERK5)与抑制剂的晶体结构
抑制剂标识:11-环戊基-2-[[2-甲氧基-4-[4-(4-甲基哌嗪-1-基)哌啶-1-基]羰基苯基]氨基]-5-甲基嘧啶并[4,5-b][1,4]苯并二氮杂䓬-6-酮
作者:Elkins, J.M、Wang, J、Vollmar, M、Mahajan, P、Savitsky, P、Deng, X、Gray, N.S、Pike, A.C.W、von Delft, F、Bountra, C、Arrowsmith, C、Edwards, A、Knapp, S
提交日期:2012-09-03
发布日期:2012-09-19
最后更新日期:2023-12-20
实验方法:X射线衍射(分辨率2.8 Å)
引用文献:《Erk5(MAPK7)与特异性抑制剂复合物的X射线晶体结构》,《J. Med. Chem.》,56卷,2013年
创建时间:
2012-09-03



