Crystal structure of human GSK3B in complex with ARN9133
收藏Protein Data Bank Japan2023-10-18 更新2026-04-19 收录
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Crystal structure of human GSK3B in complex with ARN9133 Descriptor: 3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-N,N-dimethylazetidine-1-sulfonamide, CHLORIDE ION, Glycogen synthase kinase-3 beta Authors: Tripathi, S.K, Balboni, B, Giabbai, B, Storici, P, Girotto, S, Cavalli, A. Deposit date: 2022-02-25 Release date: 2022-04-27 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Identification of Novel GSK-3 beta Hits Using Competitive Biophysical Assays. Int J Mol Sci, 23, 2022
与ARN9133结合的人源糖原合酶激酶3β(GSK3B)晶体结构
描述符:3-[2-氨基-5-(4-氟苯基)嘧啶-4-基]-N,N-二甲基氮杂环丁烷-1-磺酰胺、氯离子
作者:特里帕蒂(S.K. Tripathi)、巴洛尼(B. Balboni)、贾巴伊(B. Giabbai)、斯托里奇(P. Storici)、吉罗托(S. Girotto)、卡瓦利(A. Cavalli)
提交日期:2022-02-25
发布日期:2022-04-27
最后修改日期:2023-10-18
实验方法:X射线衍射(2.6埃)
引用文献:《利用竞争性生物物理分析法发现新型GSK-3β活性命中化合物》,刊载于《国际分子科学杂志(Int J Mol Sci)》,2022年,第23卷
创建时间:
2022-02-25



