CRYSTAL STRUCTURE OF PROTEIN TYROSINE PHOSPHATASE 1B COMPLEXED WITH TWO BIS(PARA-PHOSPHOPHENYL)METHANE (BPPM) MOLECULES
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CRYSTAL STRUCTURE OF PROTEIN TYROSINE PHOSPHATASE 1B COMPLEXED WITH TWO BIS(PARA-PHOSPHOPHENYL)METHANE (BPPM) MOLECULES Descriptor: 4-PHOSPHONOOXY-PHENYL-METHYL-[4-PHOSPHONOOXY]BENZEN, MAGNESIUM ION, PROTEIN TYROSINE PHOSPHATASE 1B Authors: Puius, Y.A, Zhao, Y, Sullivan, M, Lawrence, D, Almo, S.C, Zhang, Z.-Y. Deposit date: 1997-01-16 Release date: 1998-03-04 Last modified: 2024-05-22 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Identification of a second aryl phosphate-binding site in protein-tyrosine phosphatase 1B: a paradigm for inhibitor design. Proc.Natl.Acad.Sci.USA, 94, 1997
与双(对磷酸苯基)甲烷(BPPM)分子结合的蛋白酪氨酸磷酸酶1B的晶体结构
配体描述:4-磷酸氧基苯基-甲基-[4-磷酸氧基]苯、镁离子、蛋白酪氨酸磷酸酶1B
作者:Puius Y.A.、Zhao Y.、Sullivan M.、Lawrence D.、Almo S.C.、Zhang Z.-Y.
提交日期:1997-01-16
发布日期:1998-03-04
最后修改日期:2024-05-22
实验方法:X射线衍射(1.9 Å)
引用文献:《蛋白酪氨酸磷酸酶1B中第二个芳基磷酸酯结合位点的鉴定:抑制剂设计的范式》,美国国家科学院院刊,第94卷,1997年
创建时间:
1997-01-16



