Crystal structure of human Pim-1 kinase in complex with a consensuspeptide and (R)-3-(2-((isoquinolin-5-ylmethyl)(methyl)carbamoyl)phenyl)pyrrolidin-1-ium
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Crystal structure of human Pim-1 kinase in complex with a consensuspeptide and (R)-3-(2-((isoquinolin-5-ylmethyl)(methyl)carbamoyl)phenyl)pyrrolidin-1-ium Descriptor: Pimtide, Serine/threonine-protein kinase pim-1, ~{N}-(isoquinolin-5-ylmethyl)-~{N}-methyl-2-[(3~{R})-pyrrolidin-3-yl]benzamide Authors: Siefker, C, Heine, A, Klebe, G. Deposit date: 2017-02-14 Release date: 2018-03-07 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.21 Å) Cite: A crystallographic fragment study with human Pim-1 kinase to be published
人源Pim-1激酶与共有肽以及(R)-3-(2-((异喹啉-5-基甲基)(甲基)氨基甲酰)苯基)吡咯烷鎓的共晶结构
描述符:Pimtide、丝氨酸/苏氨酸蛋白激酶Pim-1、N-(异喹啉-5-基甲基)-N-甲基-2-[(3R)-吡咯烷-3-基]苯甲酰胺
作者:Siefker C、Heine A、Klebe G
沉积日期:2017-02-14
发布日期:2018-03-07
最后修改日期:2024-10-23
实验方法:X射线衍射(分辨率2.21 Å)
引用文献:针对人源Pim-1激酶的晶体片段研究,待发表
创建时间:
2017-02-14



