Tubulin-inhibitor complex
收藏Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6th4
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Tubulin-inhibitor complex Descriptor: 1,2,3,9-tetramethoxy-6-methylidene-5~{H}-cyclohepta[a]naphthalen-8-one, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ... Authors: Varela, P.F, Gigant, B. Deposit date: 2019-11-18 Release date: 2021-12-01 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.121 Å) Cite: B-nor-methylene Colchicinoid PT-100 Selectively Induces Apoptosis in Multidrug-Resistant Human Cancer Cells via an Intrinsic Pathway in a Caspase-Independent Manner Acs Omega, 7, 2022
微管蛋白(Tubulin)抑制剂复合物 描述符:1,2,3,9-四甲氧基-6-亚甲基-5H-环庚[a]萘-8-酮、鸟苷5'-二磷酸(Guanosine-5'-Diphosphate, GDP)、鸟苷5'-三磷酸(Guanosine-5'-Triphosphate, GTP)……
作者:Varela P.F.、Gigant B.
提交日期:2019-11-18
发布日期:2021-12-01
最后修改日期:2024-11-13
实验方法:X射线衍射(分辨率2.121 埃)
引用文献:《B-去甲亚甲基秋水仙碱类化合物PT-100通过半胱天冬酶非依赖的内源性通路选择性诱导多药耐药人癌细胞凋亡》,发表于《ACS Omega》第7卷,2022年
创建时间:
2019-11-18



