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Cryo-EM structure of human NaV1.7/beta1/beta2-TCN-1752

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Protein Data Bank Japan2025-07-02 更新2026-06-30 收录
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https://pdbj.org/mine/summary/7xmg
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Cryo-EM structure of human NaV1.7/beta1/beta2-TCN-1752 Descriptor: (1~{Z})-~{N}-[2-methyl-3-[(~{E})-[6-[4-[[4-(trifluoromethyloxy)phenyl]methoxy]piperidin-1-yl]-1~{H}-1,3,5-triazin-2-ylidene]amino]phenyl]ethanimidic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... Authors: Jiang, D.H, Zhang, J.T. Deposit date: 2022-04-25 Release date: 2022-11-30 Last modified: 2025-07-02 Method: ELECTRON MICROSCOPY (3.09 Å) Cite: Structural basis for Na V 1.7 inhibition by pore blockers. Nat.Struct.Mol.Biol., 29, 2022
创建时间:
2022-04-25
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