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crystal structures of human pyruvate dehydrogenase kinase 2 containing physiological and synthetic ligands

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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https://pdbj.org/mine/summary/2bu6
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crystal structures of human pyruvate dehydrogenase kinase 2 containing physiological and synthetic ligands Descriptor: (N-{4-[(ETHYLANILINO)SULFONYL]-2-METHYLPHENYL}-3,3,3-TRIFLUORO-2-HYDROXY-2-METHYLPROPANAMIDE, PYRUVATE DEHYDROGENASE KINASE ISOENZYME 2 Authors: Knoechel, T.R, Tucker, A.D, Robinson, C.M, Phillips, C, Taylor, W, Bungay, P.J, Kasten, S.A, Roche, T.E, Brown, D.G. Deposit date: 2005-06-08 Release date: 2006-02-02 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Regulatory Roles of the N-Terminal Domain Based on Crystal Structures of Human Pyruvate Dehydrogenase Kinase 2 Containing Physiological and Synthetic Ligands. Biochemistry, 45, 2006

含生理及合成配体的人丙酮酸脱氢酶激酶2晶体结构 描述符:(N-{4-[(乙苯胺基)磺酰基]-2-甲基苯基}-3,3,3-三氟-2-羟基-2-甲基丙酰胺)、丙酮酸脱氢酶激酶同工酶2 作者:Knoechel, T.R.、Tucker, A.D.、Robinson, C.M.、Phillips, C.、Taylor, W.、Bungay, P.J.、Kasten, S.A.、Roche, T.E.、Brown, D.G. 存储日期:2005-06-08 发布日期:2006-02-02 最后修改日期:2024-05-08 实验方法:X射线衍射(分辨率2.4埃) 引用文献:《基于含生理及合成配体的人丙酮酸脱氢酶激酶2晶体结构解析N端结构域的调控功能》,《生物化学(Biochemistry)》,2006年,第45卷
创建时间:
2005-06-08
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