Crystal structure of Klebsiella pneumoniae FabG2(NADH-dependent) at 1.57 A resolution
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Crystal structure of Klebsiella pneumoniae FabG2(NADH-dependent) at 1.57 A resolution Descriptor: 3-oxoacyl-[acyl-carrier protein] reductase, GLYCEROL, PHOSPHATE ION Authors: Vella, P, Schnell, R, Lindqvist, Y, Schneider, G. Deposit date: 2019-10-18 Release date: 2020-11-18 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.57 Å) Cite: A FabG inhibitor targeting an allosteric binding site inhibits several orthologs from Gram-negative ESKAPE pathogens. Bioorg.Med.Chem., 30, 2021
分辨率为1.57埃的肺炎克雷伯菌FabG2(NADH依赖型)晶体结构
描述项:3-氧酰基-[酰基载体蛋白]还原酶、甘油、磷酸根离子
作者:Vella P、Schnell R、Lindqvist Y、Schneider G
入库日期:2019-10-18
发布日期:2020-11-18
最后修改日期:2024-01-24
检测方法:X射线衍射(1.57 Å)
引用文献:靶向变构结合位点的FabG抑制剂可抑制革兰氏阴性ESKAPE病原体的多种同源蛋白。《Bioorg.Med.Chem.》,第30卷,2021年
创建时间:
2019-10-18



