Crystal structure of human GRP78 (70kDa heat shock protein 5 / BIP) ATPase domain in complex with ATP
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Crystal structure of human GRP78 (70kDa heat shock protein 5 / BIP) ATPase domain in complex with ATP Descriptor: 78 kDa glucose-regulated protein, ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION Authors: Dokurno, P, Surgenor, A.E, Shaw, T, Macias, A.T, Massey, A.J, Williamson, D.S. Deposit date: 2010-01-13 Release date: 2011-01-26 Last modified: 2023-09-06 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Adenosine-Derived Inhibitors of 78 kDa Glucose Regulated Protein (Grp78) ATPase: Insights into Isoform Selectivity. J.Med.Chem., 54, 2011
人类GRP78(70kDa热休克蛋白5 / BIP)ATP酶结构域与ATP结合的晶体结构
描述:78 kDa葡萄糖调节蛋白、腺苷-5'-三磷酸、镁离子
作者:Dokurno, P、Surgenor, A.E、Shaw, T、Macias, A.T、Massey, A.J、Williamson, D.S.
提交日期:2010-01-13
发布日期:2011-01-26
最后修改日期:2023-09-06
实验方法:X射线衍射(分辨率2.3 Å)
引用文献:《腺苷衍生的78 kDa葡萄糖调节蛋白(Grp78)ATP酶抑制剂:异构体选择性研究》,《药物化学杂志》(J.Med.Chem.),54卷,2011年
创建时间:
2010-01-13



