Co-crystal structure of lenacapavir bound to N74D mutant of disulfide stabilized HIV-1 CA hexamer
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Co-crystal structure of lenacapavir bound to N74D mutant of disulfide stabilized HIV-1 CA hexamer Descriptor: CAPSID PROTEIN P24, CHLORIDE ION, IODIDE ION, ... Authors: Bester, S.M, Kvaratskhelia, M. Deposit date: 2021-07-20 Release date: 2022-07-27 Last modified: 2024-12-25 Method: X-RAY DIFFRACTION (3.32 Å) Cite: Structural and Mechanistic Bases of Viral Resistance to HIV-1 Capsid Inhibitor Lenacapavir. Mbio, 13, 2022
来那卡帕韦(Lenacapavir)结合二硫键稳定的HIV-1衣壳(CA)六聚体N74D突变体的共结晶结构
描述符:衣壳蛋白P24(CAPSID PROTEIN P24)、氯离子(CHLORIDE ION)、碘离子(IODIDE ION)……
作者:Bester, S.M.、Kvaratskhelia, M.
提交日期:2021-07-20
发布日期:2022-07-27
末次修改日期:2024-12-25
实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率3.32埃(Å)
引用文献:《抗HIV-1衣壳抑制剂来那卡帕韦的病毒耐药性结构与机制基础》,Mbio,第13卷,2022年
创建时间:
2021-07-20



