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Crystal structure of c-Src in complex with covalent inhibitor LW-Srci-8

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Protein Data Bank Japan2024-10-09 更新2026-05-23 收录
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Crystal structure of c-Src in complex with covalent inhibitor LW-Srci-8 Descriptor: N-[(1R)-1-[3,5-bis(fluoranyl)phenyl]-2-(cyclopentylamino)-2-oxidanylidene-ethyl]-N-cyclopropyl-prop-2-enamide, Proto-oncogene tyrosine-protein kinase Src Authors: Zhang, H.M, Luo, C. Deposit date: 2023-06-06 Release date: 2024-06-12 Last modified: 2024-10-09 Method: X-RAY DIFFRACTION (2.724 Å) Cite: The crystal structure of c-Src in complex with covalent inhibitor LW-Srci-8 To Be Published

与共价抑制剂LW-Srci-8结合的c-Src晶体结构 描述符:N-[(1R)-1-[3,5-二氟苯基]-2-(环戊基氨基)-2-氧代乙基]-N-环丙基-2-丙烯酰胺,原癌基因酪氨酸蛋白激酶Src(Proto-oncogene tyrosine-protein kinase Src) 作者:Zhang, H.M.、Luo, C. 提交日期:2023-06-06 发布日期:2024-06-12 最后修改日期:2024-10-09 测试方法:X射线衍射(X-RAY DIFFRACTION),分辨率2.724埃 引用说明:与共价抑制剂LW-Srci-8结合的c-Src晶体结构 待发表
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2023-06-06
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