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Co-crystal Structure of Toxoplasma gondii Prolyl tRNA Synthetase (TgPRS) in complex with HFG and JE6

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Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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Co-crystal Structure of Toxoplasma gondii Prolyl tRNA Synthetase (TgPRS) in complex with HFG and JE6 Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 7-bromo-6-chloro-3-{3-[(2R,3S)-3-hydroxypiperidin-2-yl]-2-oxopropyl}quinazolin-4(3H)-one, Prolyl-tRNA synthetase (ProRS), ... Authors: Mishra, S, Malhotra, N, Manickam, Y, Sharma, A. Deposit date: 2021-05-22 Release date: 2022-03-09 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (1.697 Å) Cite: Double drugging of prolyl-tRNA synthetase provides a new paradigm for anti-infective drug development. Plos Pathog., 18, 2022

刚地弓形虫(Toxoplasma gondii)脯氨酰tRNA合成酶(TgPRS)与HFG和JE6结合的共晶体结构 数据集详情:2-(N-吗啉代)乙磺酸、7-溴-6-氯-3-{3-[(2R,3S)-3-羟基哌啶-2-基]-2-氧代丙基}喹唑啉-4(3H)-酮、脯氨酰-tRNA合成酶(Prolyl-tRNA synthetase, ProRS)…… 作者:Mishra S、Malhotra N、Manickam Y、Sharma A 提交日期:2021-05-22 发布日期:2022-03-09 最后修改日期:2023-11-29 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率1.697埃(Å) 引用文献:《双重靶向脯氨酰-tRNA合成酶为抗感染药物开发提供新范式》,发表于《公共科学图书馆·病原体》(Plos Pathog.),2022年,第18卷
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2021-05-22
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