Kinetics, stability, and structural changes in high resolution crystal structures of HIV-1 protease with drug resistant mutations L24I, I50V, AND G73S
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Kinetics, stability, and structural changes in high resolution crystal structures of HIV-1 protease with drug resistant mutations L24I, I50V, AND G73S Descriptor: DIMETHYL SULFOXIDE, GLYCEROL, N-{(2S)-2-[(N-acetyl-L-threonyl-L-isoleucyl)amino]hexyl}-L-norleucyl-L-glutaminyl-N~5~-[amino(iminio)methyl]-L-ornithinamide, ... Authors: Liu, F, Boross, P.I, Wang, Y.F, Tozser, J, Louis, J.M, Harrison, R.W, Weber, I.T. Deposit date: 2005-08-30 Release date: 2006-01-24 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (1.3 Å) Cite: Kinetic, stability, and structural changes in high-resolution crystal structures of HIV-1 protease with drug-resistant mutations L24I, I50V, and G73S. J.Mol.Biol., 354, 2005
携带耐药突变L24I、I50V及G73S的HIV-1蛋白酶高分辨率晶体结构的动力学、稳定性与结构变化
描述符:二甲基亚砜(DIMETHYL SULFOXIDE)、甘油(GLYCEROL)、N-{(2S)-2-[(N-乙酰基-L-苏氨酰-L-异亮氨酰)氨基]己基}-L-正亮氨酰-L-谷氨酰胺基-N~5~-[氨基(亚氨基鎓)甲基]-L-鸟氨酰胺,……
作者:Liu, F、Boross, P.I、Wang, Y.F、Tozser, J、Louis, J.M、Harrison, R.W、Weber, I.T
提交日期:2005-08-30
发布日期:2006-01-24
最后修改日期:2024-03-13
实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率1.3埃(Å)
引用文献:《携带耐药突变L24I、I50V及G73S的HIV-1蛋白酶高分辨率晶体结构的动力学、稳定性与结构变化》,《分子生物学杂志》(J.Mol.Biol.),第354卷,2005年
创建时间:
2005-08-30



